SCHEMBL8305023

SCHEMBL8305023

CC(=O)Nc1ccc2c(CCC(=O)O)c(C(=O)c3ccncc3)oc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
KDM4E B2RXH2 7/20 0.44
HPGD P15428 7/20 0.44
HSD17B10 Q99714 6/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
GLA P06280 2/20 0.40
GAA P10253 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAP2K1 Q02750 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
TSHR P16473 4/20 0.39
MAPT P10636 2/20 0.38
RAB9A P51151 1/20 0.38
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305025 0.92 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8307013 0.88 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL8326272 0.86 CA12 (0.41) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL8837860 0.82 KDM4E (0.52) ALDH1A1KDM4EHPGDHSD17B10GLA
SCHEMBL8553130 0.81 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8324883 0.81 NPC1 (0.48) ALDH1A1KDM4EHSD17B10LMNASMN1; SMN2
SCHEMBL8307015 0.79 KDM4E (0.46) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL9075776 0.78 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9070589 0.78 CA12 (0.43) ALDH1A1KDM4EHPGDSMN1; SMN2CA12
SCHEMBL8554638 0.76 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685475-B1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1999-01-13 EP disclosed
EP-0685474-B1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1998-09-16 EP disclosed
US-5622989-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
US-5565488-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
EP-0685475-A1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed
EP-0685474-A1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed