SCHEMBL8305025

SCHEMBL8305025

CC(=O)Nc1ccc2oc(C(=O)c3ccncc3)c(CCC(=O)O)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.41
TSHR P16473 5/20 0.41
KDM4E B2RXH2 7/20 0.41
HPGD P15428 4/20 0.41
HSD17B10 Q99714 4/20 0.41
MAPT P10636 4/20 0.41
MAPK1 P28482 3/20 0.41
ALOX15 P16050 2/20 0.41
PKM P14618 1/20 0.41
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.39
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 2/20 0.37
ELANE P08246 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305023 0.92 ALDH1A1 (0.44) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8307015 0.88 KDM4E (0.46) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8553140 0.81 MAPT (0.39) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8307013 0.79 ALDH1A1 (0.45) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8326272 0.78 CA12 (0.41) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL9070592 0.78 KDM4E (0.45) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8554644 0.76 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL8837860 0.76 KDM4E (0.52) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8841212 0.75 ALDH1A1 (0.46) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL8553130 0.75 ALDH1A1 (0.38) ALDH1A1TSHRKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685475-B1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1999-01-13 EP disclosed
US-5622989-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0685475-A1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed