SCHEMBL8306246

SCHEMBL8306246

COc1ccccc1C(=O)c1cccn1NC(=O)CN

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.47
NPC1 O15118 2/20 0.45
LMNA P02545 3/20 0.42
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC1 Q13547 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39
GLA P06280 1/20 0.39
STS P08842 1/20 0.39
STAT3 P40763 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8307230 0.99 CTSD (0.46) CTSDNPC1LMNAALOX15HSD17B10
SCHEMBL8441148 0.81 GABRP (0.48) NPC1LMNAHSD17B10KMT2AMEN1
SCHEMBL9122774 0.80 HDAC1 (0.43) CTSDNPC1LMNAHDAC1KMT2A
Bromide SCHEMBL8305746 0.80 CES2 (0.37) NPC1ALOX15KMT2AMEN1HPGD
Hydrochloric Acid SCHEMBL8304040 0.80 GABRP (0.47) NPC1LMNAHSD17B10KMT2AMEN1
Bromide SCHEMBL10365922 0.80 CES2 (0.37) NPC1ALOX15KMT2AMEN1HPGD
Bromide SCHEMBL8305743 0.80 CES2 (0.37) NPC1ALOX15KMT2AMEN1HPGD
Bromide SCHEMBL10367565 0.80 GABRP (0.47) NPC1LMNAHSD17B10KMT2AMEN1
SCHEMBL8304637 0.79 NPC1 (0.48) NPC1LMNAALOX15KMT2AMEN1
SCHEMBL8308215 0.78 LMNA (0.41) LMNAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582182-B1 1-Aminoacetamidopyrroles and 1-amino-2-(substituted) pyrroles and their use for the treatment of neurodegenerative dysfunctions HOECHST MARION ROUSSEL INC (US) 1999-10-20 EP claimed
US-5428053-A Treats alzheimer's disease and other senile dementias HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-06-27 US claimed