SCHEMBL8306747

SCHEMBL8306747

N=C(Nc1ccc2c(c1)CCC2NCc1ccccc1)C1=CC=CCC1=S

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
GRIN2B Q13224 2/20 0.34
NPY1R P25929 7/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
PLA2G1B P04054 1/20 0.33
HPGD P15428 1/20 0.33
MAOB P27338 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308398 0.88 KMT2A (0.37) KDM4EALDH1A1MAOB
SCHEMBL8306856 0.87 KDM4E (0.43) KDM4EALDH1A1
SCHEMBL8310235 0.84 GRIN2B (0.49) GRIN2B
SCHEMBL8309546 0.81 FYN (0.47) GRIN2B
SCHEMBL8307046 0.77 KDM1A (0.48) KDM4EGRIN2BALDH1A1MAOB
SCHEMBL8305839 0.77 GRIN2B (0.38) GRIN2B
SCHEMBL8309243 0.76 MTTP (0.45)
SCHEMBL8177517 0.76 ACKR3 (0.40) KDM4EGRIN2BALDH1A1LMNAMAOB
SCHEMBL8309227 0.75 DRD2 (0.40) GRIN2BLMNA
SCHEMBL8306217 0.74 SMO (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759027-B1 BICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHETASE ASTRA AB (SE) 1999-08-04 EP claimed