SCHEMBL8307686

SCHEMBL8307686

O=C(Nc1cccc2ccccc12)c1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.68
CHEK1 O14757 1/20 0.61
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
KMT2A Q03164 4/20 0.58
MEN1 O00255 3/20 0.58
MAPT P10636 6/20 0.56
ALDH1A1 P00352 3/20 0.56
POLB P06746 1/20 0.56
LMNA P02545 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
RORC P51449 1/20 0.55
SIRT6 Q8N6T7 1/20 0.54
HTT P42858 1/20 0.54
HCAR3 P49019 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026664 0.89 MAPT (0.67) ALOX5CHEK1KMT2AMEN1MAPT
SCHEMBL9232842 0.82 ALOX5 (0.78) ALOX5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL8306313 0.80 AKR1C2 (0.65) CHEK1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL6900995 0.80 CYP1A2 (0.63) ALOX5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL8305753 0.79 SMN1; SMN2 (0.74) NPC1RAB9ACYP1A2CYP3A4CYP2C9
SCHEMBL18992223 0.79 ALOX5 (0.72) ALOX5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL21914836 0.78 NPC1 (0.80) ALOX5NPC1RAB9ACYP1A2CYP3A4
SCHEMBL8308004 0.78 MEN1 (0.69) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL8445659 0.78 LMNA (0.71) NPC1RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL12113016 0.78 ALOX5 (0.73) ALOX5NPC1RAB9ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934068-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-08-11 EP disclosed
WO-1998009630-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1998-03-12 WO disclosed