SCHEMBL8308037

SCHEMBL8308037

Cc1ccc(N)cc1OC(C)c1ncc[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
GAA P10253 2/20 0.35
ADRA2A P08913 3/20 0.33
ADRA2B P18089 3/20 0.33
ADRA2C P18825 3/20 0.33
NISCH Q9Y2I1 2/20 0.33
CASP1 P29466 2/20 0.33
RECQL P46063 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
F7 P08709 1/20 0.32
P2RX3 P56373 1/20 0.32
P2RX2 Q9UBL9 1/20 0.32
F2RL1 P55085 2/20 0.31
CYP3A4 P08684 2/20 0.31
TSHR P16473 2/20 0.31
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309503 0.82 POLB (0.45) ALDH1A1GAAADRA2AADRA2BADRA2C
SCHEMBL11189892 0.74 ADRA2A (0.40) ALDH1A1GAAADRA2AADRA2BADRA2C
SCHEMBL8145073 0.71 ALDH1A1 (0.48) ALDH1A1GAACASP1RECQLKDM4E
Hydrochloric Acid SCHEMBL9756776 0.70 ALDH1A1 (0.46) ALDH1A1GAANISCHCASP1RECQL
SCHEMBL15651168 0.69 NISCH (0.46) ALDH1A1GAAADRA2ANISCHCASP1
SCHEMBL3633273 0.69 SMPD3 (0.50) ALDH1A1GAANISCHKDM4EMAPT
SCHEMBL11691601 0.69 CASP1 (0.45) ALDH1A1GAACASP1RECQLKDM4E
SCHEMBL10370479 0.68 KDM4E (0.50) ADRA2AADRA2BADRA2CNISCHKDM4E
SCHEMBL2968176 0.68 MAOB (0.39) ADRA2AADRA2BADRA2CCYP3A4
SCHEMBL11689564 0.67 TDP1 (0.56) ALDH1A1GAACASP1RECQLKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed