SCHEMBL8308890

SCHEMBL8308890

O=C1CCc2cccc(OCCCCN3CCCN(Cc4ccc5ccccc5n4)CC3)c2N1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.49
HTR1A P08908 8/20 0.46
HTR2A P28223 8/20 0.46
DRD1 P21728 1/20 0.45
DRD4 P21917 1/20 0.45
DRD5 P21918 1/20 0.45
HTR2C P28335 1/20 0.45
DRD3 P35462 1/20 0.45
HTR2B P41595 1/20 0.45
MAOA P21397 3/20 0.44
MAOB P27338 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310251 0.97 DRD2 (0.46) DRD2HTR1AHTR2ADRD1DRD4
SCHEMBL6584872 0.97 DRD2 (0.48) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6586928 0.95 MAOA (0.45) DRD2HTR1AHTR2ADRD4DRD3
SCHEMBL6585890 0.84 DRD2 (0.43) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6586944 0.83 MAOA (0.58) DRD2HTR1AHTR2ADRD4HTR2C
SCHEMBL6587330 0.83 DRD2 (0.43) DRD2HTR1AHTR2AMAOAMAOB
SCHEMBL6584969 0.83 MAOA (0.67) DRD2MAOAMAOB
SCHEMBL6585295 0.83 MAOA (0.59) DRD2HTR1AHTR2ADRD4HTR2C
SCHEMBL6585490 0.82 MAOA (0.68) DRD2MAOAMAOB
SCHEMBL6584734 0.82 HTR1A (0.41) DRD2HTR1AHTR2AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed