SCHEMBL8309375

SCHEMBL8309375

O=C(NCc1ccco1)[C@H](Cc1ccccc1)NC(=O)[C@H]1N[C@@H]1C(=O)O.[NaH]

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.52
PSMB5 P28074 1/20 0.52
PSMB2 P49721 1/20 0.52
ALDH1A1 P00352 6/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
TSHR P16473 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
CTSL P07711 1/20 0.48
BRS3 P32247 1/20 0.47
HTT P42858 1/20 0.46
MAPT P10636 3/20 0.46
MAPK1 P28482 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.45
RECQL P46063 1/20 0.43
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309378 0.89 PSMB1 (0.50) PSMB1PSMB5PSMB2ALDH1A1MEN1
SCHEMBL8309254 0.86 PSMB1 (0.49) PSMB1PSMB5PSMB2ALDH1A1MEN1
SCHEMBL7354817 0.83 PSMB1 (0.52) PSMB1PSMB5PSMB2ALDH1A1MEN1
SCHEMBL7355264 0.83 MMP1 (0.47) MEN1KMT2ABRS3
SCHEMBL7358942 0.82 KMT2A (0.53) PSMB1PSMB5PSMB2MEN1KMT2A
SCHEMBL7354151 0.81 CTSL (0.46) CTSL
SCHEMBL7361514 0.81 BACE1 (0.48) PSMB5ALDH1A1MEN1KMT2ACTSL
SCHEMBL7362211 0.81 MCHR1 (0.47) MEN1KMT2A
SCHEMBL7356263 0.81 TSHR (0.56) ALDH1A1KMT2ATSHRCTSLHTT
SCHEMBL7361179 0.80 MME (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753003-B1 AZIRIDINE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-06-16 EP disclosed
US-5668128-A INHIBITORS OF THIOL PROTEASE, PROPHYLAXIS AND TREATMENT OF BONE DISEASES, OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-09-16 US disclosed