SCHEMBL8309535

SCHEMBL8309535

COc1cc(N)c(Cl)cc1-c1nn(C2CCN(CCc3ccccc3)CC2)c(=O)o1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.44
DRD2 P14416 5/20 0.43
DRD3 P35462 5/20 0.43
ACHE P22303 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRK1 P41145 1/20 0.43
HTR2B P41595 1/20 0.43
CHRNA4 P43681 1/20 0.43
HTR3A P46098 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310238 0.86 DRD4 (0.48) DRD4DRD2DRD3
SCHEMBL8305104 0.85 HTR4 (0.44) HTR4
Hydrochloric Acid SCHEMBL8368070 0.84 HTR4 (0.43) HTR4
SCHEMBL8309549 0.82 ACHE (0.51) ACHEHTR4
SCHEMBL6961633 0.81 HTR4 (0.47) ACHECYP2D6CYP2C9KCNH2HTR4
Capeserod SCHEMBL4707724 0.80 HTR4 (0.45) DRD2CYP3A4CYP1A2ADRA2ACYP2D6
Bromide SCHEMBL7744560 0.80 HTR4 (0.46) ACHECYP2D6CYP2C9KCNH2HTR4
Capeserod SCHEMBL399091 0.80 HTR4 (0.44) DRD2DRD3ADRA2AADRA2CHTR2A
SCHEMBL8304880 0.79 HTR4 (0.44) ACHEHTR3AHTR4
Bromide SCHEMBL8366387 0.78 HTR4 (0.43) ACHEHTR3AHTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929089-A ANTISEROTONINE AGENT SYNTHELABO (FR) 1999-07-27 US disclosed
EP-0863897-B1 5-PHENYL-3-(PIPERIDIN-4-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES FOR USE AS 5-HT4- OR H3-RECEPTOR LIGANDS SYNTHELABO (FR) 1999-06-16 EP disclosed