SCHEMBL8312609

SCHEMBL8312609

CCC(=O)c1cc(F)cnc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.39
KCNH2 Q12809 1/20 0.38
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
HSP90AB1 P08238 1/20 0.36
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HMGCR P04035 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.32
CHRNA7 P36544 1/20 0.32
APLNR P35414 1/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
PTGS1 P23219 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9928617 0.80 AGBL2 (0.39) AGBL2KCNH2SCN5ASCN9ASMN1; SMN2
SCHEMBL27734476 0.79 HSP90AB1 (0.36) HSP90AB1ALDH1A1SMN1; SMN2HMGCRKDM4E
SCHEMBL2086658 0.79 CASP1 (0.47) ALDH1A1SMN1; SMN2L3MBTL1TSHRKMT2A
SCHEMBL27598069 0.78 KEAP1 (0.53) AGBL2SCN5ASCN9AALDH1A1SMN1; SMN2
SCHEMBL31349524 0.78 KEAP1 (0.53) AGBL2SCN5ASCN9AALDH1A1SMN1; SMN2
SCHEMBL290570 0.78 KEAP1 (0.53) AGBL2SCN5ASCN9AALDH1A1SMN1; SMN2
SCHEMBL4966985 0.78 ALDH1A1 (0.36) AGBL2SCN5ASCN9AALDH1A1SMN1; SMN2
SCHEMBL8357219 0.78 SCN5A (0.36) AGBL2SCN5ASCN9ASMN1; SMN2KMT2A
SCHEMBL27286638 0.77 ALDH1A1 (0.38) AGBL2SCN5ASCN9AALDH1A1KMT2A
SCHEMBL168694 0.77 CASP1 (0.42) SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009966-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed