SCHEMBL8312241

SCHEMBL8312241

O=C1c2c(c3c4ccccc4[nH]c3c3[nH]c4ccccc4c23)C(=O)N1Cc1ccccn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.66
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 2/20 0.55
HSD17B10 Q99714 1/20 0.55
PRKCA P17252 4/20 0.55
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
PKM P14618 1/20 0.54
CDK4 P11802 5/20 0.51
CCND1 P24385 5/20 0.51
CYP1B1 Q16678 1/20 0.50
PRKD3 O94806 2/20 0.48
PRKCG P05129 2/20 0.48
PRKCB P05771 2/20 0.48
PRKACA P17612 2/20 0.48
PRKACG P22612 2/20 0.48
PRKACB P22694 2/20 0.48
PRKCH P24723 2/20 0.48
PRKCI P41743 2/20 0.48
PRKCE Q02156 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313203 0.80 NQO1 (1.00) NQO1ALDH1A1KDM4EPRKCAMEN1
SCHEMBL13431714 0.77 NQO1 (0.73) NQO1ALDH1A1KDM4EHSD17B10PRKCA
SCHEMBL20624192 0.74 PRKD3 (0.61) NQO1HSD17B10PRKCACDK4CCND1
SCHEMBL8324352 0.72 NQO1 (0.74) NQO1KDM4EPRKCAMEN1KMT2A
SCHEMBL9374032 0.72 SIRT2 (0.66) ALDH1A1KDM4EHSD17B10PRKCAMEN1
SCHEMBL8317372 0.71 PRKCA (1.00) NQO1PRKCAMEN1KMT2ACDK4
SCHEMBL5438544 0.71 PRKCA (0.71) NQO1PRKCAMEN1KMT2ACDK4
SCHEMBL4095113 0.71 ALDH1A1 (0.64) ALDH1A1KDM4EHSD17B10MEN1KMT2A
Hydrochloric Acid SCHEMBL8319377 0.71 SIRT2 (0.64) ALDH1A1KDM4EHSD17B10PRKCAMEN1
SCHEMBL30711693 0.71 ALDH1A1 (1.00) ALDH1A1KDM4EHSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP claimed
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP disclosed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US disclosed