SCHEMBL8313240

SCHEMBL8313240

CC1(C)C=C(c2ccccn2)c2ccc(C(F)(F)F)cc2OC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 2/20 0.35
TGFBR1 P36897 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PDK2 Q15119 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MDM2 Q00987 1/20 0.34
DRD2 P14416 1/20 0.34
GRM5 P41594 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312741 0.91 CBFB (0.39) CBFBSMN1; SMN2NPC1MAPK1RAB9A
SCHEMBL8315309 0.82 ADRA1A (0.38) SMN1; SMN2NPC1RAB9ALMNAMAPT
SCHEMBL8311146 0.82 ABCC9 (0.34) CBFBTGFBR1PDK2KCNH2
SCHEMBL8316184 0.81 KDM4E (0.37) SMN1; SMN2NPC1MAPK1RAB9AGAA
SCHEMBL8311427 0.81 SCN9A (0.35) CBFBMAPK1RAB9AALDH1A1LMNA
SCHEMBL8313018 0.79 METAP2 (0.39) TGFBR1ALDH1A1MEN1MAPTKMT2A
SCHEMBL8316296 0.78 CCR1 (0.35) SMN1; SMN2NPC1MAPK1RAB9AALDH1A1
SCHEMBL8314584 0.77 FABP6 (0.37) CBFBRAB9ATGFBR1MAPTGRM5
SCHEMBL8315666 0.77 NTRK1 (0.35) NPC1RAB9AALDH1A1MAPTGRM5
SCHEMBL8315603 0.76 CBFB (0.42) CBFBGRM5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed