SCHEMBL8310381

SCHEMBL8310381

CC1(C)C=C(c2ccccn2)c2cc(-c3ccccc3)ccc2OC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.40
TMEM97 Q5BJF2 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
HTR7 P34969 1/20 0.40
HTR1A P08908 1/20 0.39
PGR P06401 2/20 0.38
MAPT P10636 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
TP53 P04637 2/20 0.36
PKM P14618 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
KLF5 Q13887 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 2/20 0.36
POLB P06746 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315486 0.85 NPC1 (0.39) PGRMAPTRAB9ASMN1; SMN2TP53
SCHEMBL8315585 0.84 ADRA1A (0.40) PGRMAPTRAB9ASMN1; SMN2TP53
SCHEMBL8312863 0.84 MAPT (0.39) PGRMAPTRAB9ASMN1; SMN2TP53
SCHEMBL8314584 0.84 FABP6 (0.37) PGRMAPTRAB9ATGFBR1BACE1
SCHEMBL8316184 0.83 KDM4E (0.37) HTR7MAPTRAB9ASMN1; SMN2TP53
SCHEMBL8313611 0.82 NPC1 (0.41) HTR2BTMEM97SIGMAR1HTR7HTR1A
SCHEMBL8314548 0.82 NPC1 (0.35) MAPTRAB9ASMN1; SMN2TP53PKM
SCHEMBL8310538 0.82 GABRA1 (0.34) MAPTRAB9ASMN1; SMN2TP53PKM
SCHEMBL8312741 0.81 CBFB (0.39) MAPTRAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8313790 0.81 TGFBR1 (0.39) MAPTKDM4EALDH1A1TSHRTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed