SCHEMBL8313843

SCHEMBL8313843

O=C(Nc1ccc(C(=O)O)c(Cl)c1)c1cc(F)ccc1F

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.61
OXTR P30559 1/20 0.61
AVPR1A P37288 1/20 0.61
PYGL P06737 3/20 0.55
NPC1 O15118 6/20 0.52
RAB9A P51151 6/20 0.52
FADS1 O60427 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
GRM4 Q14833 1/20 0.51
PNLIP P16233 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
MAPT P10636 2/20 0.49
ANO1 Q5XXA6 1/20 0.48
ANO2 Q9NQ90 1/20 0.48
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GRIK1 P39086 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331533 0.86 AVPR2 (0.79) AVPR2OXTRAVPR1APYGLNPC1
SCHEMBL22871324 0.83 AVPR2 (0.55) AVPR2OXTRAVPR1APYGLNPC1
SCHEMBL7341264 0.81 TSHR (0.68) AVPR2PYGLNPC1RAB9ATDP1
SCHEMBL27316696 0.80 AVPR2 (0.54) AVPR2OXTRAVPR1ANPC1RAB9A
SCHEMBL8317450 0.80 NPC1 (0.65) AVPR2OXTRAVPR1ANPC1RAB9A
SCHEMBL8316833 0.78 SMN1; SMN2 (0.61) PYGLNPC1RAB9AMAPTSMN1; SMN2
SCHEMBL12700230 0.78 ALDH1A1 (0.64) AVPR2OXTRAVPR1ANPC1RAB9A
SCHEMBL1197393 0.78 PYGL (0.64) AVPR2OXTRAVPR1APYGLNPC1
SCHEMBL7334964 0.77 AVPR2 (0.57) AVPR2OXTRAVPR1ANPC1RAB9A
SCHEMBL7824838 0.77 FADS1 (0.72) NPC1RAB9AFADS1NPSR1PNLIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed
CN-1039908-C Tricyclic diaza * vasopressin antagonists and oxytocin antagonists AMERICAN CYANAMID CO (US) 1998-09-23 CN disclosed