SCHEMBL8314007

SCHEMBL8314007

O=C1Cc2c(ccc3c2OC(CNCc2ccc(F)cc2)CC3)N1

nearest known ligand 0.81

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.81
DRD4 P21917 6/20 0.81
DRD3 P35462 6/20 0.81
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
SLC6A4 P31645 6/20 0.44
HTR2A P28223 2/20 0.42
HTR2B P41595 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312627 0.90 DRD2 (0.81) DRD2DRD4DRD3NFKB1NFKB2
SCHEMBL8314369 0.90 DRD2 (0.81) DRD2DRD4DRD3NFKB1NFKB2
SCHEMBL8312005 0.90 DRD2 (1.00) DRD2DRD4DRD3NFKB1NFKB2
SCHEMBL8313970 0.87 DRD2 (0.77) DRD2DRD4DRD3NFKB1NFKB2
SCHEMBL5957081 0.82 DRD2 (0.55) DRD2DRD4DRD3SLC6A4HTR2A
SCHEMBL8314765 0.79 DRD2 (0.68) DRD2DRD4DRD3NFKB1NFKB2
SCHEMBL8643128 0.77 DRD2 (0.64) DRD2DRD4DRD3SLC6A4HTR2A
SCHEMBL8317510 0.77 DRD2 (0.64) DRD2DRD4DRD3SLC6A4HTR2A
SCHEMBL7395323 0.72 DRD2 (0.45) DRD2DRD4DRD3SLC6A4HTR2A
SCHEMBL5957139 0.71 DRD2 (0.55) DRD2DRD4DRD3SLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP claimed
EP-0771801-B1 Chromane derivatives AMERICAN HOME PROD (US) 1999-03-03 EP claimed
EP-0771801-A1 Chromane derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1997-05-07 EP claimed
EP-0771801-B1 Chromane derivatives AMERICAN HOME PROD (US) 1999-03-03 EP disclosed
EP-0771801-A1 Chromane derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1997-05-07 EP disclosed