SCHEMBL8314864

SCHEMBL8314864

CSc1ccc2c(c1)C(O)(c1ccccn1)CC(C)(C)CO2

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.37
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
GRM4 Q14833 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316835 0.85 SLC6A2 (0.39) SLC6A2NPC1RAB9A
SCHEMBL8311266 0.85 SLC6A2 (0.37) SLC6A2
SCHEMBL8311974 0.84 BACE1 (0.37) SLC6A2SMN1; SMN2
SCHEMBL8313637 0.84 SLC6A2 (0.36) SLC6A2NPC1RAB9A
SCHEMBL8310708 0.83 SLC6A2 (0.40) SLC6A2SMN1; SMN2
SCHEMBL8314119 0.83 HTR2B (0.38) SLC6A2NPC1RAB9ASMN1; SMN2
SCHEMBL8313905 0.82 PDK2 (0.35) SLC6A2RAB9A
SCHEMBL8314935 0.82 SCN9A (0.38) SLC6A2NPC1RAB9ASMN1; SMN2
SCHEMBL8313766 0.82 PDK2 (0.35) SLC6A2
SCHEMBL8313558 0.81 SLC6A2 (0.38) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed