SCHEMBL8314577

SCHEMBL8314577

Clc1ccc(-c2ccccc2C=C2CCNCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
HTR2C P28335 6/20 0.39
HTR2A P28223 5/20 0.39
HTR2B P41595 4/20 0.39
HTR7 P34969 3/20 0.38
HTR6 P50406 2/20 0.38
HTR3A P46098 1/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
HTR1D P28221 1/20 0.37
HTR1E P28566 1/20 0.37
PRCP P42785 1/20 0.36
HTR1A P08908 1/20 0.36
CHRM2 P08172 1/20 0.36
PTGS2 P35354 2/20 0.35
PTGS1 P23219 1/20 0.35
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314716 0.84 HTR7 (0.48) HTR2CHTR2AHTR2BHTR7HTR6
SCHEMBL8313295 0.84 CHRM1 (0.55) HTR2CHTR2AHTR2BHTR7CHRM1
Hydrochloric Acid SCHEMBL10600743 0.83 HTR7 (0.47) HTR2CHTR2AHTR2BHTR7HTR6
SCHEMBL1497170 0.81 CYP26A1 (0.39) PTGS2PTGS1CYP1A2
SCHEMBL8316750 0.81 HTR1A (0.51) HTR2CHTR2AHTR2BHTR7HTR1A
SCHEMBL12751389 0.76 DYRK2 (0.51) HTR2CHTR2AHTR2BHTR7
Hydrochloric Acid SCHEMBL7983894 0.75 DYRK2 (0.50) HTR2CHTR2AHTR2BHTR7
Hydrochloric Acid SCHEMBL10601953 0.73 HTR7 (0.42) HTR2CHTR2AHTR2BHTR7HTR6
SCHEMBL8316880 0.73 HRH3 (0.39) SIGMAR1HTR2CHTR2AHTR2BHTR7
SCHEMBL16322736 0.72 HTR2C (0.48) SIGMAR1HTR2CHTR2AHTR2BHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed