SCHEMBL8315438

SCHEMBL8315438

COc1ccc(-c2ccccc2C=C2CCN(CCCCl)CC2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
TMEM97 Q5BJF2 1/20 0.40
DRD2 P14416 3/20 0.39
DRD4 P21917 3/20 0.39
DRD3 P35462 3/20 0.39
ABCB1 P08183 4/20 0.39
ABCC1 P33527 1/20 0.38
QPCT Q16769 1/20 0.38
BACE1 P56817 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316861 0.86 HRH3 (0.48) KCNH2HRH3BACE1
SCHEMBL8312632 0.85 ABCB1 (0.47) KCNH2HRH3SIGMAR1TMEM97DRD2
SCHEMBL8317603 0.82 HRH3 (0.40) HRH3SIGMAR1DRD3BACE1
SCHEMBL8316880 0.81 HRH3 (0.39) HRH3SIGMAR1DRD2DRD3
SCHEMBL8314770 0.80 CHRM1 (0.40) KCNH2HRH3
SCHEMBL8316992 0.80 HRH3 (0.39) KCNH2HRH3DRD2DRD4DRD3
SCHEMBL8312305 0.79 MC4R (0.39) KCNH2HRH3BACE1
SCHEMBL8316497 0.77 MC4R (0.39) KCNH2HRH3DRD2DRD3
SCHEMBL10559968 0.75 KCNH2 (0.49) KCNH2HRH3SIGMAR1DRD2DRD4
Oxalic Acid SCHEMBL10558317 0.73 ALDH1A1 (0.50) KCNH2SIGMAR1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed