SCHEMBL8312632

SCHEMBL8312632

COc1cccc(-c2ccccc2C=C2CCN(CCCCl)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
HTR7 P34969 2/20 0.44
DRD4 P21917 3/20 0.43
DRD3 P35462 3/20 0.43
DRD2 P14416 2/20 0.43
BACE1 P56817 1/20 0.42
HRH3 Q9Y5N1 2/20 0.42
HTR1A P08908 3/20 0.41
SIGMAR1 Q99720 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2C P28335 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
HTR2B P41595 1/20 0.41
SLC6A3 Q01959 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316861 0.88 HRH3 (0.48) HTR7BACE1HRH3HTR1AKCNH2
SCHEMBL8315438 0.85 KCNH2 (0.43) ABCB1ABCC1DRD4DRD3DRD2
SCHEMBL8314770 0.84 CHRM1 (0.40) HTR7HRH3HTR1ACHRM3SLC6A3
SCHEMBL8317603 0.82 HRH3 (0.40) DRD3BACE1HRH3SIGMAR1
SCHEMBL8316880 0.78 HRH3 (0.39) HTR7DRD3DRD2HRH3HTR1A
SCHEMBL8316992 0.78 HRH3 (0.39) HTR7DRD4DRD3DRD2HRH3
SCHEMBL8312305 0.77 MC4R (0.39) BACE1HRH3CHRM3KCNH2ALDH1A1
SCHEMBL8316497 0.75 MC4R (0.39) DRD3DRD2HRH3ADRA1DADRA1A
SCHEMBL11037599 0.69 HTR7 (0.41) HTR7DRD3DRD2BACE1HRH3
Hydrochloric Acid SCHEMBL11034929 0.69 HTR7 (0.41) HTR7DRD3DRD2BACE1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed