SCHEMBL8316014

SCHEMBL8316014

CCOC(=O)c1cc(NC)c(C)nc1C(=O)OCC

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
ALOX15 P16050 1/20 0.56
KDM4E B2RXH2 3/20 0.52
HPGD P15428 1/20 0.52
MAPT P10636 4/20 0.48
GAA P10253 1/20 0.48
KMT2A Q03164 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
POLB P06746 1/20 0.46
TSHR P16473 2/20 0.45
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323222 0.85 ALDH1A1 (0.62) ALDH1A1ALOX15KDM4EHPGDMAPT
SCHEMBL9800425 0.84 KDM4E (0.50) ALDH1A1ALOX15KDM4EHPGDGAA
SCHEMBL9315414 0.78 SMN1; SMN2 (0.56) ALDH1A1ALOX15KDM4EHPGDMAPT
SCHEMBL8322828 0.78 KDM4E (0.51) ALDH1A1ALOX15KDM4EHPGDMAPT
SCHEMBL8661094 0.78 ALDH1A1 (0.50) ALDH1A1ALOX15KDM4EHPGDMAPT
SCHEMBL9205477 0.77 TSHR (0.49) ALDH1A1ALOX15KDM4EHPGDGAA
SCHEMBL9316182 0.75 KDM4E (0.44) ALDH1A1ALOX15KDM4EHPGDGAA
SCHEMBL9315811 0.75 ALOX15 (0.45) ALDH1A1ALOX15KDM4EHPGDGAA
SCHEMBL9316161 0.74 KDM4E (0.43) ALDH1A1ALOX15KDM4EHPGDGAA
SCHEMBL8661697 0.74 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5959116-A 5-NITRO PYRIDINE-2,3-DICARBOXYLIC ACID ESTER CHEMICAL INTERMEDIATES MADE BY REACTING THE N-OXIDES OF PYRIDINE-2,3-DICARBOXYLIC ACID ESTERS WITH NITRIC ACID OR SODIUM NITRATE, THEN REMOVING THE N-OXIDE GROUP BASF AKTIENGESELLSCHAFT (DE) 1999-09-28 US claimed
EP-0663399-B1 Pyridine-2,3-dicarboxylic imides, process for their preparation and their use to control the growth of unwanted plants BASF AG (DE) 1998-06-10 EP claimed
US-5959116-A 5-NITRO PYRIDINE-2,3-DICARBOXYLIC ACID ESTER CHEMICAL INTERMEDIATES MADE BY REACTING THE N-OXIDES OF PYRIDINE-2,3-DICARBOXYLIC ACID ESTERS WITH NITRIC ACID OR SODIUM NITRATE, THEN REMOVING THE N-OXIDE GROUP BASF AKTIENGESELLSCHAFT (DE) 1999-09-28 US disclosed
US-5571774-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1996-11-05 US disclosed