SCHEMBL8316079

SCHEMBL8316079

COc1ccc(Cn2c(C)cc3c(=O)[nH][nH]c(=O)c32)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.57
ALDH1A1 P00352 2/20 0.53
MAPT P10636 2/20 0.53
KDM4E B2RXH2 2/20 0.53
ALOX15 P16050 1/20 0.53
PDE1B Q01064 6/20 0.48
PDE1C Q14123 6/20 0.48
PDE1A P54750 5/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
P2RX4 Q99571 1/20 0.47
PIK3R1 P27986 2/20 0.46
PIK3CA P42336 2/20 0.46
CMA1 P23946 1/20 0.45
RXFP1 Q9HBX9 1/20 0.44
DAO P14920 1/20 0.44
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313452 0.83 ALDH1A1 (0.56) TYMSALDH1A1MAPTKDM4EMEN1
SCHEMBL4769071 0.76 ALDH1A1 (0.60) TYMSALDH1A1MAPTKDM4EALOX15
SCHEMBL8312892 0.74 TYMS (0.58) TYMSALDH1A1MAPTKDM4EALOX15
SCHEMBL8315901 0.74 ALDH1A1 (0.54) TYMSALDH1A1MAPTKDM4EALOX15
SCHEMBL26988574 0.73 MAPT (0.49) ALDH1A1MAPTKDM4EALOX15PDE1B
SCHEMBL31560451 0.71 MAPT (0.72) ALDH1A1MAPTKDM4EALOX15PDE1B
SCHEMBL4376098 0.70 ALDH1A1 (0.57) TYMSALDH1A1MAPTKDM4EALOX15
SCHEMBL17675021 0.70 ALDH1A1 (0.57) TYMSALDH1A1MAPTKDM4EALOX15
SCHEMBL8924914 0.70 KDM4E (1.00) ALDH1A1MAPTKDM4EALOX15MEN1
SCHEMBL4762572 0.70 ALDH1A1 (0.63) TYMSALDH1A1MAPTKDM4EALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609328-B1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-28 EP disclosed
US-5534515-A Pyrrolopyridazines having gastrointestinal protective effects BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-07-09 US disclosed
WO-1993008190-A1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-04-29 WO disclosed