SCHEMBL8315901

SCHEMBL8315901

COc1ccc(Cn2c(C)cc3c(Cl)nnc(Cl)c32)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
MAPT P10636 3/20 0.54
KDM4E B2RXH2 2/20 0.54
ALOX15 P16050 1/20 0.54
DCTPP1 Q9H773 3/20 0.50
TYMS P04818 1/20 0.49
PDE1B Q01064 6/20 0.46
PDE1C Q14123 6/20 0.46
PDE1A P54750 5/20 0.46
GAA P10253 1/20 0.43
GFER P55789 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
P2RX4 Q99571 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
LMNA P02545 1/20 0.41
CNR2 P34972 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312429 0.83 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EALOX15TYMS
SCHEMBL8316587 0.83 ALDH1A1 (0.50) ALDH1A1MAPTKDM4EALOX15DCTPP1
SCHEMBL8316729 0.82 ALDH1A1 (0.50) ALDH1A1MAPTKDM4ETYMSKMT2A
SCHEMBL8313591 0.80 DCTPP1 (0.50) ALDH1A1MAPTKDM4EALOX15DCTPP1
SCHEMBL2475307 0.76 ALDH1A1 (0.51) ALDH1A1MAPTKDM4EALOX15DCTPP1
SCHEMBL8316079 0.74 TYMS (0.57) ALDH1A1MAPTKDM4EALOX15TYMS
SCHEMBL22270343 0.73 MAPT (0.51) ALDH1A1MAPTKDM4EALOX15DCTPP1
SCHEMBL8924914 0.71 KDM4E (1.00) ALDH1A1MAPTKDM4EALOX15DCTPP1
SCHEMBL8459060 0.71 DYRK1A (0.43) ALDH1A1MAPTKDM4ETYMSL3MBTL1
SCHEMBL8314143 0.71 DYRK1A (0.43) ALDH1A1MAPTKDM4ETYMSKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609328-B1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-28 EP disclosed
US-5534515-A Pyrrolopyridazines having gastrointestinal protective effects BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-07-09 US disclosed
WO-1993008190-A1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-04-29 WO disclosed