SCHEMBL8317200

SCHEMBL8317200

CCOC(=O)c1ccc(NC(=O)c2cccc(Cl)c2Cl)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.54
CYP1A2 P05177 1/20 0.54
ALDH1A1 P00352 4/20 0.51
POLB P06746 2/20 0.51
KDM4E B2RXH2 2/20 0.51
PKM P14618 1/20 0.51
GAA P10253 2/20 0.48
NPC1 O15118 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
F2R P25116 1/20 0.48
MITF O75030 1/20 0.47
WDR5 P61964 1/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
TDP1 Q9NUW8 2/20 0.46
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319324 0.90 RAB9A (0.64) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8316866 0.87 RAB9A (0.56) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL7334998 0.87 ALDH1A1 (0.65) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8315129 0.85 WDR5 (0.52) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8318448 0.84 ALDH1A1 (0.56) RAB9ACYP1A2ALDH1A1KDM4EGAA
SCHEMBL6961250 0.83 ALDH1A1 (0.54) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8317169 0.83 ALDH1A1 (0.67) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8316571 0.82 HDAC1 (0.57) RAB9ACYP1A2ALDH1A1KDM4ENPC1
SCHEMBL8319329 0.82 RAB9A (0.53) RAB9ACYP1A2ALDH1A1POLBKDM4E
SCHEMBL8318097 0.82 CYP1A2 (0.55) RAB9ACYP1A2ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed