SCHEMBL8317634

SCHEMBL8317634

CCOC(=O)OC1CC(OC)CN1C(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
DPP4 P27487 1/20 0.39
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.38
ERCC1 P07992 1/20 0.38
ERCC4 Q92889 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
P2RX7 Q99572 2/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
RECQL P46063 1/20 0.36
ADCY8 P40145 1/20 0.36
MEN1 O00255 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317448 0.90 KMT2A (0.40) KMT2ADPP4LMNASMN1; SMN2TSHR
SCHEMBL8312980 0.90 KMT2A (0.40) KMT2ADPP4LMNASMN1; SMN2TSHR
SCHEMBL8312982 0.86 OPRK1 (0.35) KMT2ADPP4SMN1; SMN2TSHRP2RX7
SCHEMBL8318856 0.84 KMT2A (0.40) KMT2ADPP4LMNASMN1; SMN2TSHR
SCHEMBL8875871 0.84 TSHR (0.41) KMT2ADPP4LMNASMN1; SMN2TSHR
SCHEMBL8314255 0.84 CYP3A4 (0.35) KMT2ALMNASMN1; SMN2P2RX7CYP3A4
SCHEMBL8317694 0.84 KMT2A (0.43) KMT2ALMNASMN1; SMN2TSHRERCC1
SCHEMBL8318785 0.83 KMT2A (0.43) KMT2ADPP4SMN1; SMN2TSHRSIGMAR1
SCHEMBL9538321 0.82 SIGMAR1 (0.49) KMT2ATSHRSIGMAR1PDE3BPDE3A
SCHEMBL9386772 0.81 KMT2A (0.40) KMT2ADPP4LMNASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501129-B1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1999-07-14 EP disclosed
EP-0501129-A1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1992-09-02 EP disclosed