SCHEMBL8317854

SCHEMBL8317854

COc1ccc(C(=C2CCN(CCCCl)CC2)c2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
DRD3 P35462 2/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 1/20 0.43
SIGMAR1 Q99720 3/20 0.43
ACHE P22303 1/20 0.42
PRSS1 P07477 3/20 0.41
EBP Q15125 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HTR1A P08908 1/20 0.40
HTR2A P28223 1/20 0.40
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315432 0.94 OPRM1 (0.48) CYP2D6CYP2C9KMT2AMEN1DRD3
SCHEMBL8316856 0.79 OPRM1 (0.52) DRD3DRD2SIGMAR1HTR1AHTR2A
SCHEMBL8312626 0.78 DRD4 (0.47) KMT2ADRD2DRD4SIGMAR1ALDH1A1
SCHEMBL8315004 0.78 OPRD1 (0.47)
SCHEMBL8313011 0.78 DRD2 (0.45) CYP2D6CYP2C9KMT2AMEN1DRD3
SCHEMBL10557192 0.78 DRD3 (0.51) DRD3DRD2SMN1; SMN2ALDH1A1HPGD
SCHEMBL10462690 0.78 KMT2A (0.49) KMT2AMEN1DRD3DRD2DRD4
SCHEMBL27508978 0.77 OPRM1 (0.45) KMT2AMEN1DRD3DRD2DRD4
SCHEMBL10559361 0.76 KMT2A (0.57) KMT2AMEN1DRD3DRD2DRD4
SCHEMBL10460413 0.76 KDM4E (0.50) KMT2AMEN1DRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
US-5683998-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, ANTIPAF AGENTS TORAY INDUSTRIES, INC. (JP) 1997-11-04 US disclosed