SCHEMBL8317984

SCHEMBL8317984

NC(=O)c1cn(C2Cc3ccccc3C2=O)c(C(N)=O)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ACHE P22303 5/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
NOTUM Q6P988 1/20 0.35
BCAT2 O15382 1/20 0.34
METAP1 P53582 4/20 0.33
CYP19A1 P11511 1/20 0.33
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32
HTR2B P41595 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317672 0.93 SMN1; SMN2 (0.37) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL8643929 0.87 ACHE (0.34) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL8316817 0.84 SMN1; SMN2 (0.40) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL8555113 0.79 KDM4E (0.40) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL8649980 0.77 GABRA2 (0.45) MEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8316162 0.75 MAPT (0.41) MEN1MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL8650346 0.73 MAPT (0.39) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL8316058 0.71 KMO (0.37) ACHEHTR2BHTR2C
SCHEMBL8558771 0.69 KDM4E (0.40) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL10821600 0.68 ACHE (0.40) KDM4EMEN1MAPTKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772615-B1 IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-2-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE POULENC RORER SA (FR) 1999-09-22 EP disclosed
US-5726175-A MULTISTAGE PROCESS WITH CYCLIZATION AND AMINATION RHONE-POULENC RORER S.A. (FR) 1998-03-10 US disclosed
EP-0772615-A1 IMIDAZO 1,2-a]INDENO 1,2-e]PYRAZINE-2-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1997-05-14 EP disclosed
WO-1996002544-A1 IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-2-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1996-02-01 WO disclosed