SCHEMBL8317985

SCHEMBL8317985

CC(C)(C)OC(=O)c1ccc(CCc2ccccc2OCc2ccccc2)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.46
DRD2 P14416 4/20 0.46
PTGER1 P34995 2/20 0.42
PTGER4 P35408 2/20 0.42
PTGER3 P43115 2/20 0.42
PTGER2 P43116 2/20 0.42
ABCB1 P08183 9/20 0.42
HTT P42858 1/20 0.39
ABCG2 Q9UNQ0 2/20 0.38
FOLH1 Q04609 1/20 0.38
LMNA P02545 1/20 0.38
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8321520 0.88 CCR5 (0.46) PTGER1HTTLMNA
SCHEMBL8326795 0.86 HTR1A (0.54) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL9056586 0.85 MEN1 (0.44)
SCHEMBL8675704 0.74 HDAC3 (0.44) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8324470 0.74 PTGER1 (0.48) PTGER1HTTFOLH1LMNA
SCHEMBL8321988 0.73 HTR1A (0.52) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8162190 0.73 CCR5 (0.44) PTGER1HTTLMNA
SCHEMBL8324638 0.71 MRGPRX4 (0.44) PTGER1FOLH1
SCHEMBL19511860 0.71 PTGER1 (0.49) PTGER1HTT
SCHEMBL4429436 0.71 KDM4E (0.53) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed