SCHEMBL8317991

SCHEMBL8317991

O=[C]c1c(F)cccc1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.37
GAA P10253 1/20 0.35
RAB9A P51151 5/20 0.33
NPC1 O15118 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PTGS2 P35354 1/20 0.33
KIF11 P52732 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.31
VNN1 O95497 1/20 0.31
CXCL8 P10145 1/20 0.30
PSIP1 O75475 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989031 0.74 NFE2L2 (0.37) KCNN4GAARAB9ANPC1SMN1; SMN2
SCHEMBL6993867 0.71 CES1 (0.43) KCNN4GAARAB9ANPC1SMN1; SMN2
SCHEMBL95707 0.70 CES2 (0.42) ALDH1A1
SCHEMBL6989492 0.66 CES2 (0.37) KCNN4GAARAB9ANPC1SMN1; SMN2
SCHEMBL15941518 0.65 KIF11 (0.39) KCNN4GAARAB9ASMN1; SMN2KIF11
SCHEMBL7705802 0.63 CES2 (0.36) ALDH1A1
SCHEMBL163604 0.62 SLC22A12 (0.38) GAASMN1; SMN2PTGS2ALDH1A1
SCHEMBL21201383 0.61 ACHE (0.48) GAAKMT2AALDH1A1
SCHEMBL7156428 0.61 CES2 (0.39) GAARAB9ANPC1SMN1; SMN2MEN1
SCHEMBL535572 0.61 TAAR1 (0.41) GAASMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929533-A1 4,4-DISUBSTITUTED-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONES USEFUL AS HIV REVERSE TRANSCRIPTASE INHIBITORS AND INTERMEDIATES AND PROCESSES FOR MAKING THE SAME Du Pont Pharmaceuticals Company (US) 1999-07-21 EP disclosed
WO-1998014436-A1 4,4-DISUBSTITUTED-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONES USEFUL AS HIV REVERSE TRANSCRIPTASE INHIBITORS AND INTERMEDIATES AND PROCESSES FOR MAKING THE SAME DUPONT PHARMACEUTICALS COMPANY (US) 1998-04-09 WO disclosed