SCHEMBL8318035

SCHEMBL8318035

CCCCOC(=O)N1CCCC(O)C1c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.40
HTR7 P34969 1/20 0.38
GBA2 Q9HCG7 1/20 0.38
HTR2A P28223 1/20 0.38
FKBP1A P62942 3/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
SLC10A2 Q12908 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059786 0.88 CHRM2 (0.46) KMT2AMEN1L3MBTL1GBA2FKBP1A
SCHEMBL9274408 0.88 CHRM2 (0.46) KMT2AMEN1L3MBTL1GBA2FKBP1A
SCHEMBL8154541 0.79 MEN1 (0.43) KMT2AMEN1MAPK1HTTHTR7
SCHEMBL6668590 0.76 CHRM2 (0.45) KMT2AMEN1L3MBTL1FKBP1AKDM4E
SCHEMBL932669 0.74 RIPK1 (0.46) HCRTR2
SCHEMBL2731646 0.73 POLB (0.46) KMT2AMEN1L3MBTL1GBA2FKBP1A
SCHEMBL4202768 0.73 POLB (0.46) KMT2AMEN1L3MBTL1GBA2FKBP1A
SCHEMBL31421713 0.73 LMNA (0.47) KMT2AMEN1L3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL17674467 0.73 GBA2 (0.44) L3MBTL1GBA2ALDH1A1SMN1; SMN2CHRM2
SCHEMBL29747664 0.71 GCK (0.40) L3MBTL1FKBP1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906315-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1999-04-07 EP disclosed
WO-1997049710-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1997-12-31 WO disclosed
EP-0683767-A1 AZACYCLIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1995-11-29 EP disclosed
WO-1994019323-A1 AZACYCLIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1994-09-01 WO disclosed