SCHEMBL8319129

SCHEMBL8319129

CS(=O)(=O)OC1CN2C3CC(NC(=O)c4c[nH]c5ccccc45)CC2CC1C3

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.52
HTR3E A5X5Y0 4/20 0.52
HTR3B O95264 4/20 0.52
HTR3D Q70Z44 4/20 0.52
HTR3C Q8WXA8 4/20 0.52
KCNH2 Q12809 4/20 0.49
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA7 P36544 2/20 0.41
CHRNA4 P43681 2/20 0.41
SLC6A4 P31645 2/20 0.41
HTR4 Q13639 2/20 0.41
CHRNA1 P02708 1/20 0.41
CHRNG P07510 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM5 P08912 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319125 1.00 HTR3A (0.52) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8319559 0.85 KCNH2 (0.62) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8323177 0.82 KCNH2 (0.68) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8323170 0.82 KCNH2 (0.68) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9705203 0.81 HTR3A (0.53) HTR3ANR4A2
SCHEMBL8320783 0.80 HTR3A (0.41) HTR3AKCNH2CYP3A4
SCHEMBL8323360 0.77 ALDH1A1 (0.61) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8323356 0.77 ALDH1A1 (0.61) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9471661 0.75 HTR3A (0.71) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL13186221 0.75 HTR3A (0.85) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955470-A Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed