SCHEMBL8320783

SCHEMBL8320783

CS(=O)(=O)OC1CN2C3CC(NC(=O)c4cccc5c4oc4ccccc45)CC2CC1C3

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 16/20 0.41
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
KCNH2 Q12809 2/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319125 0.80 HTR3A (0.52) HTR3AKCNH2CYP3A4
SCHEMBL9705203 0.80 HTR3A (0.53) HTR3A
SCHEMBL8319129 0.80 HTR3A (0.52) HTR3AKCNH2CYP3A4
SCHEMBL8323360 0.75 ALDH1A1 (0.61) HTR3AKCNH2CYP3A4
SCHEMBL8323356 0.75 ALDH1A1 (0.61) HTR3AKCNH2CYP3A4
SCHEMBL9706213 0.70 HTR3A (0.33) HTR3AKCNH2
SCHEMBL8320785 0.65 KCNH2 (0.37) KCNH2
SCHEMBL8319559 0.65 KCNH2 (0.62) HTR3AKCNH2CYP3A4
SCHEMBL516118 0.64 ALOX5 (0.52) HDAC1HDAC8HDAC6
SCHEMBL976167 0.64 HDAC8 (0.59) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955470-A Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed