SCHEMBL8319658

SCHEMBL8319658

COc1ccc2[nH]c(C)c(C3=C(c4c(Cc5cccc(CN)c5)[nH]c5ccccc45)C(=O)NC3=O)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.45
CAMK2D Q13557 3/20 0.42
ABCG2 Q9UNQ0 1/20 0.41
CCNE1 P24864 2/20 0.40
CDK2 P24941 2/20 0.40
CCNE2 O96020 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CAMK2B Q13554 1/20 0.40
CAMK2G Q13555 1/20 0.40
CAMK2A Q9UQM7 1/20 0.40
PRKCB P05771 2/20 0.39
PRKCA P17252 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
HTR1D P28221 1/20 0.39
HTR6 P50406 1/20 0.39
PDGFRB P09619 1/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317092 1.00 ROCK2 (0.45) ROCK2CAMK2DABCG2CCNE1CDK2
Hydrochloric Acid SCHEMBL8319262 0.99 ROCK2 (0.44) ROCK2CAMK2DABCG2CCNE1CDK2
SCHEMBL8318394 0.96 HTR6 (0.42) ROCK2ABCG2MTNR1AMTNR1BHTR1D
SCHEMBL8317078 0.91 CAMK2D (0.48) CAMK2DCDK4CCND1CAMK2BCAMK2G
Hydrochloric Acid SCHEMBL8318720 0.90 CAMK2D (0.48) CAMK2DCDK4CCND1CAMK2BCAMK2G
Hydrochloric Acid SCHEMBL8316493 0.86 CAMK2D (0.42) CAMK2DCCNE1CDK2CCNE2CDK4
SCHEMBL8314912 0.84 PRKCB (0.42) CAMK2DPRKCBPRKCAMEN1KMT2A
SCHEMBL8316483 0.84 CAMK2D (0.51) CAMK2DPRKCBPRKCAGSK3BCHEK1
SCHEMBL8314832 0.82 CAMK2D (0.43) CAMK2DCDK4CCND1CAMK2BCAMK2G
Hydrochloric Acid SCHEMBL8317707 0.81 CAMK2D (0.42) CAMK2DCDK4CCND1CAMK2BCAMK2G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925296-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS Astra Aktiebolag (SE) 1999-06-30 EP disclosed
WO-1998011102-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRA AKTIEBOLAG (SE) 1998-03-19 WO disclosed