SCHEMBL8320138

SCHEMBL8320138

CN1CCN(c2ccc(Cl)c(C(F)(F)F)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.59
NOTUM Q6P988 12/20 0.52
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HSD17B10 Q99714 1/20 0.50
PHGDH O43175 1/20 0.50
DPP4 P27487 2/20 0.48
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20080888 0.92 NOTUM (0.58) NOTUMMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL8320134 0.84 NOTUM (0.52) NOTUMMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL2922525 0.84 DPP4 (0.52) NOTUMMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL2921346 0.83 DPP4 (0.51) NOTUMMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL21448004 0.82 SIRT6 (0.61) SIRT6MEN1KMT2ASMN1; SMN2
SCHEMBL9645889 0.82 MAPT (0.50) NOTUMMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL3243736 0.81 NOTUM (0.53) SIRT6NOTUMMEN1CYP1A2CYP3A4
SCHEMBL30340643 0.81 GAA (0.61) SIRT6MEN1KMT2ASMN1; SMN2
SCHEMBL255333 0.81 ADRB1 (0.65) NOTUMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL13068417 0.81 GAA (0.61) SIRT6MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
EP-2508526-A1 Spiroalkene carboxamide derivatives and their use as chemokine receptor modulators Ares Trading SA (CH) 2012-10-10 EP disclosed
WO-2012130915-A1 SPIROALKENE CARBOXAMIDE DERIVATIVES AND THEIR USE AS CHEMOKINE RECEPTOR MODULATORS ARES TRADING S.A. (CH) 2012-10-04 WO disclosed
US-5945421-A TREATING PSYCHOSIS AND SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1999-08-31 US disclosed