SCHEMBL8320735

SCHEMBL8320735

CC(C)(C)OC(=O)C1CCC2(CCn3c(cc4ccccc43)C2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.39
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
USP30 Q70CQ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327015 0.72 CYP11B2 (0.53) SIGMAR1USP30
SCHEMBL8326656 0.69 CYP11B2 (0.48) SIGMAR1USP30
SCHEMBL8325900 0.69 HTR2A (0.46) SIGMAR1HTR2AHTR2C
SCHEMBL8328249 0.69 HTR2A (0.44) SIGMAR1HTR2AHTR2C
SCHEMBL6590757 0.68 KCNA3 (0.50) SIGMAR1
SCHEMBL8325258 0.67 CYP11B2 (0.53) SIGMAR1USP30
SCHEMBL615033 0.66 SIGMAR1 (0.63) SIGMAR1
SCHEMBL8325766 0.66 CRBN (0.46) HTR2AHTR2C
SCHEMBL6715677 0.66 HTR2A (0.53) SIGMAR1HTR2AHTR2C
SCHEMBL3542987 0.66 NOTUM (0.40) SIGMAR1BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed