SCHEMBL8320869

SCHEMBL8320869

C=CCN(C(=O)OCCCC)c1cccc(CO)c1I

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.35
TDP1 Q9NUW8 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HPGD P15428 3/20 0.34
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
ESR1 P03372 3/20 0.32
ALDH1A1 P00352 3/20 0.32
MAPK1 P28482 3/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
MCL1 Q07820 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207086 0.81 L3MBTL1 (0.33) TSHRL3MBTL1MEN1KMT2AHPGD
SCHEMBL11419708 0.69 TDP1 (0.35) TSHRTDP1L3MBTL1MEN1KMT2A
SCHEMBL6205322 0.67 TSHR (0.34) TSHRL3MBTL1
SCHEMBL28021915 0.67 TSHR (0.49) TSHRMEN1KMT2AALDH1A1RAB9A
SCHEMBL10797117 0.66 CA12 (0.41) TSHRL3MBTL1MEN1KMT2AALDH1A1
SCHEMBL27728586 0.65 TSHR (0.57) TSHRTDP1L3MBTL1HPGDESR1
SCHEMBL20297003 0.64 L3MBTL1 (0.35) TSHRTDP1L3MBTL1MEN1KMT2A
SCHEMBL11635872 0.64 ALDH1A1 (0.56) TSHRTDP1L3MBTL1ALDH1A1MAPK1
SCHEMBL12676660 0.64 GABRA1 (0.50) ALDH1A1LMNA
SCHEMBL11546490 0.63 TSHR (0.50) TSHRTDP1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938474-A2 CYCLOPROPYLINDOLE COMPOUNDS AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-09-01 EP disclosed
WO-1998011101-A2 CONDENSED N-ACLYINDOLES AS ANTITUMOR AGENTS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1998-03-19 WO disclosed