SCHEMBL8322937

SCHEMBL8322937

COC(=O)/C=C/c1ccc(Cn2cnc(-c3ccccc3)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP2E1 P05181 1/20 0.49
CYP2A6 P11509 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2B6 P20813 1/20 0.49
HPGDS O60760 1/20 0.47
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
IP6K1 Q92551 1/20 0.45
IP6K3 Q96PC2 1/20 0.45
IP6K2 Q9UHH9 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KDM4C Q9H3R0 2/20 0.44
KDM5A P29375 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
HDAC1 Q13547 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326744 0.87 HDAC1 (0.56) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8325813 0.87 TBXAS1 (0.56) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8324714 0.82 CA12 (0.48) CYP3A4CYP2D6CYP2C19KMT2AKDM4E
SCHEMBL8169471 0.82 CDK5 (0.45) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8169470 0.82 CDK5 (0.45) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL3439436 0.80 MEN1 (0.59) KMT2ANPC1RAB9AHDAC1HDAC8
SCHEMBL8323972 0.79 BRD4 (0.43) KMT2AKDM4ESMN1; SMN2IP6K1IP6K3
SCHEMBL8319688 0.78 TBXAS1 (0.46) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8325909 0.78 HDAC4 (0.55) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8318730 0.77 TBXAS1 (0.60) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed