SCHEMBL8326744

SCHEMBL8326744

O=C(/C=C/c1ccc(Cn2cnc(-c3ccccc3)c2)cc1)NO

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.56
HDAC8 Q9BY41 8/20 0.56
HDAC2 Q92769 8/20 0.55
HDAC3 O15379 6/20 0.52
CYP2E1 P05181 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2A6 P11509 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
HDAC6 Q9UBN7 8/20 0.52
HDAC4 P56524 6/20 0.52
HDAC7 Q8WUI4 4/20 0.51
HDAC10 Q969S8 4/20 0.51
HDAC11 Q96DB2 4/20 0.51
HDAC9 Q9UKV0 4/20 0.51
HDAC5 Q9UQL6 4/20 0.51
KCNH2 Q12809 1/20 0.51
HPGDS O60760 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325813 0.90 TBXAS1 (0.56) HDAC1HDAC8HDAC2HDAC3CYP2E1
SCHEMBL8325909 0.90 HDAC4 (0.55) HDAC1HDAC8HDAC2HDAC3CYP2E1
SCHEMBL8322937 0.87 CYP3A4 (0.49) HDAC1HDAC8CYP2E1CYP3A4CYP2D6
SCHEMBL8319264 0.80 HDAC6 (0.54) HDAC1HDAC8HDAC2HDAC3HDAC6
SCHEMBL8318730 0.80 TBXAS1 (0.60) CYP2E1CYP3A4CYP2D6CYP2A6CYP2C9
SCHEMBL3439437 0.79 MEN1 (0.62) HDAC1HDAC8HDAC2HDAC3HDAC6
SCHEMBL1346083 0.77 HPGDS (0.77) CYP2E1CYP3A4CYP2D6CYP2A6CYP2C9
SCHEMBL8324956 0.77 HDAC1 (0.54) HDAC1HDAC8HDAC2HDAC3HDAC6
SCHEMBL8319277 0.75 HDAC1 (0.55) HDAC1HDAC8HDAC2HDAC3HDAC6
SCHEMBL5758431 0.75 HPGDS (0.64) CYP2E1CYP3A4CYP2D6CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed