SCHEMBL8325813

SCHEMBL8325813

O=C(O)/C=C/c1ccc(Cn2cnc(-c3ccccc3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C19 P33261 2/20 0.56
USP2 O75604 1/20 0.56
LMNA P02545 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CYP2E1 P05181 1/20 0.54
CYP2A6 P11509 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2B6 P20813 1/20 0.54
HPGDS O60760 1/20 0.52
KDM4C Q9H3R0 3/20 0.48
KDM5A P29375 2/20 0.48
KDM5B Q9UGL1 2/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326744 0.90 HDAC1 (0.56) CYP3A4CYP2D6CYP2C19CYP2E1CYP2A6
SCHEMBL8318730 0.89 TBXAS1 (0.60) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8322937 0.87 CYP3A4 (0.49) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8325909 0.82 HDAC4 (0.55) TBXAS1CYP3A4CYP2D6CYP2C19CYP2E1
SCHEMBL8170143 0.80 CYP19A1 (0.48) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8170145 0.80 CYP19A1 (0.48) TBXAS1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL1346083 0.79 HPGDS (0.77) CYP3A4CYP2D6CYP2C19LMNACYP2E1
SCHEMBL3439435 0.78 MEN1 (0.65) MEN1KMT2ANPC1RAB9AGAA
SCHEMBL5758431 0.77 HPGDS (0.64) CYP3A4CYP2D6CYP2C19LMNAMEN1
SCHEMBL8319688 0.76 TBXAS1 (0.46) TBXAS1CYP3A4CYP2D6CYP2C19CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed