SCHEMBL8323370

SCHEMBL8323370

COc1cc(-c2nnn[nH]2)ccc1CCc1ccccc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 18/20 0.50
HTR1A P08908 3/20 0.50
DRD2 P14416 3/20 0.50
ABCG2 Q9UNQ0 2/20 0.50
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
NPY1R P25929 1/20 0.43
HTT P42858 1/20 0.43
NPY2R P49146 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325042 0.96 ABCB1 (0.46) ABCB1HTR1ADRD2ABCG2KDM4E
SCHEMBL8322255 0.90 ABCB1 (0.43) ABCB1HTR1ADRD2ABCG2KDM4E
SCHEMBL8321903 0.87 HTR1A (0.48) ABCB1HTR1ADRD2ABCG2
SCHEMBL8408170 0.85 HTR1A (0.61) ABCB1HTR1ADRD2ABCG2
SCHEMBL8320664 0.85 HTR1A (0.61) ABCB1HTR1ADRD2ABCG2
SCHEMBL8323974 0.83 HTR1A (0.43) ABCB1HTR1ADRD2ABCG2
SCHEMBL1247768 0.82 TSHR (0.50) KDM4ELMNAKMT2ASMN1; SMN2
SCHEMBL8325617 0.81 PTGER1 (0.55) ABCB1HTR1ADRD2ABCG2HTT
SCHEMBL8406776 0.80 ABCB1 (0.55) ABCB1HTR1ADRD2ABCG2
SCHEMBL8409574 0.76 HTR1A (0.45) ABCB1HTR1ADRD2ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP claimed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP claimed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO claimed
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed