SCHEMBL8324285

SCHEMBL8324285

N#Cc1cc2n(c1-c1cccnc1Cl)CCC=C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.34
CNR2 P34972 3/20 0.32
CNR1 P21554 2/20 0.32
PDE4A P27815 1/20 0.32
ALDH1A1 P00352 2/20 0.31
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
RECQL P46063 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964888 0.77 CYP11B2 (0.32) CYP11B2ALDH1A1MAPTKDM4ENPC1
SCHEMBL7965413 0.77 NPC1 (0.32) CYP11B2ALDH1A1KDM4ENPC1RAB9A
SCHEMBL7962248 0.76 CYP11B2 (0.31) CYP11B2
SCHEMBL7962898 0.74 ALDH1A1 (0.32) ALDH1A1MAPTKDM4ERAB9A
SCHEMBL8328943 0.74 CNR2 (0.36) CYP11B2CNR2CNR1PDE4AKDM4E
SCHEMBL8326860 0.73 NPC1 (0.34) MAPTKDM4ENPC1RAB9AMEN1
SCHEMBL7967502 0.73 GAA (0.32) ALDH1A1MAPTKDM4ERECQLRAB9A
SCHEMBL7964706 0.72 KDM4E (0.33) CYP11B2ALDH1A1MAPTKDM4E
SCHEMBL8329854 0.71 DHODH (0.36) ALDH1A1MAPTKDM4ERAB9A
SCHEMBL7952832 0.71 HCRTR1 (0.34) ALDH1A1MAPTKDM4ERAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP disclosed
US-5908863-A ANTIGROWTH AGENT FOR BONES DOMPE' S.P.A. (IT) 1999-06-01 US disclosed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO disclosed