SCHEMBL8324364

SCHEMBL8324364

CNC(NCC1CCCN(Cc2ccncc2)C1)=C(C#N)C#N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
POLB P06746 3/20 0.42
MEN1 O00255 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
BCHE P06276 1/20 0.42
NPC1 O15118 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
BLM P54132 1/20 0.41
ACKR3 P25106 1/20 0.41
LMNA P02545 2/20 0.40
GAA P10253 2/20 0.40
PKM P14618 1/20 0.40
CCR1 P32246 1/20 0.39
CCR3 P51677 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326146 0.88 TP53 (0.48) KMT2APOLBMEN1BCHEALDH1A1
SCHEMBL8326334 0.88 KMT2A (0.56) KMT2APOLBMEN1BCHEALDH1A1
SCHEMBL8330451 0.87 ALDH1A1 (0.49) KMT2APOLBMEN1BCHEALDH1A1
SCHEMBL8327677 0.86 POLB (0.54) KMT2APOLBMEN1NPC1ALDH1A1
SCHEMBL8329545 0.85 CCR3 (0.53) KMT2APOLBMEN1ALDH1A1GAA
SCHEMBL8330706 0.84 KMT2A (0.52) KMT2APOLBMEN1BCHEALDH1A1
SCHEMBL8329014 0.81 POLB (0.61) KMT2APOLBMEN1ALDH1A1LMNA
SCHEMBL7495142 0.80 ALDH1A1 (0.41) KMT2AMEN1CYP1A2CYP3A4CYP2C9
SCHEMBL8324359 0.77 MAPT (0.44) KMT2APOLBMEN1CYP1A2CYP3A4
SCHEMBL8324361 0.76 CYP1A2 (0.40) KMT2APOLBMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed