SCHEMBL8326146

SCHEMBL8326146

CNC(NCC1CCCN(Cc2ccc(Cl)cc2)C1)=C(C#N)C#N

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.48
LTA4H P09960 1/20 0.46
KMT2A Q03164 4/20 0.45
POLB P06746 3/20 0.45
MEN1 O00255 2/20 0.45
GAA P10253 2/20 0.44
BCHE P06276 1/20 0.42
CYP2D6 P10635 1/20 0.41
ACKR3 P25106 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CCR2 P41597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326334 0.91 KMT2A (0.56) KMT2APOLBMEN1GAABCHE
SCHEMBL8329545 0.90 CCR3 (0.53) KMT2APOLBMEN1GAAALDH1A1
SCHEMBL8327677 0.89 POLB (0.54) KMT2APOLBMEN1GAAALDH1A1
SCHEMBL8324364 0.88 KMT2A (0.42) KMT2APOLBMEN1GAABCHE
SCHEMBL8330451 0.88 ALDH1A1 (0.49) KMT2APOLBMEN1GAABCHE
SCHEMBL8330706 0.87 KMT2A (0.52) LTA4HKMT2APOLBMEN1GAA
SCHEMBL8329014 0.84 POLB (0.61) KMT2APOLBMEN1GAAALDH1A1
SCHEMBL7498333 0.80 DRD4 (0.53) CYP2D6
SCHEMBL8326114 0.77 MEN1 (0.48) KMT2AMEN1
SCHEMBL8326148 0.75 LTA4H (0.45) TP53LTA4HKMT2APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed