SCHEMBL8327558

SCHEMBL8327558

CCCCCC1C(C(=O)O)=C(C)NC(c2cccnc2)=C1C(=O)OCC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.54
TRPV1 Q8NER1 3/20 0.53
MAPT P10636 2/20 0.50
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 4/20 0.44
CACNA1C Q13936 1/20 0.44
NPSR1 Q6W5P4 3/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2D6 P10635 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TMIGD3 P0DMS9 1/20 0.44
GAA P10253 3/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327248 0.88 ADORA3 (0.68) ADORA3TRPV1ALDH1A1TMIGD3HPGD
SCHEMBL8324841 0.80 ADORA3 (0.46) ADORA3TRPV1MAPTMAPK1ALDH1A1
SCHEMBL8325950 0.79 ADORA3 (0.46) ADORA3TRPV1MAPTALDH1A1CYP3A4
SCHEMBL8330375 0.78 ADORA3 (0.42) ADORA3TRPV1
SCHEMBL8328228 0.77 ADORA3 (0.44) ADORA3TRPV1MAPTMAPK1ALDH1A1
SCHEMBL8323291 0.75 ADORA3 (0.43) ADORA3TRPV1
SCHEMBL29173860 0.74 ALDH1A1 (0.71) ADORA3TRPV1MAPTALDH1A1MEN1
SCHEMBL1665260 0.74 MAPT (0.68) ADORA3MAPTMAPK1ALDH1A1CACNA1C
SCHEMBL8797106 0.73 LMNA (0.49) TRPV1MAPTALDH1A1MEN1KMT2A
SCHEMBL8797103 0.73 LMNA (0.51) MAPTALDH1A1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0943615-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 1999-09-22 EP disclosed