SCHEMBL8324955

SCHEMBL8324955

COC(=O)c1ccc(CCc2cc(OC)ccc2OCc2ccccc2)cc1O

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.59
MTNR1B P49286 6/20 0.59
ABCB1 P08183 5/20 0.55
HTR1A P08908 2/20 0.54
DRD2 P14416 2/20 0.54
APP P05067 1/20 0.49
TSHR P16473 1/20 0.48
MAOB P27338 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319605 0.92 MTNR1A (0.58) MTNR1AMTNR1BABCB1HTR1ADRD2
SCHEMBL8321603 0.88 PTGER1 (0.54) MTNR1AMTNR1BABCB1HTR1ADRD2
SCHEMBL8319729 0.88 ABCB1 (0.56) ABCB1HTR1ADRD2MAOB
SCHEMBL8322935 0.88 CCR5 (0.49)
SCHEMBL8327489 0.85 LMNA (0.43) MTNR1AMTNR1BABCB1HTR1ADRD2
SCHEMBL8324057 0.82 PTGER4 (0.59) MTNR1AMTNR1BABCB1HTR1ADRD2
SCHEMBL11557673 0.81 KDM4E (0.60) MTNR1AMTNR1BAPPMAOB
SCHEMBL8406718 0.80 ABCB1 (0.63) MTNR1AMTNR1BABCB1HTR1ADRD2
SCHEMBL6258777 0.79 HSP90AA1 (0.50) TSHR
SCHEMBL8325289 0.79 ABCB1 (0.62) MTNR1AMTNR1BABCB1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed