SCHEMBL8325472

SCHEMBL8325472

CS(=O)(=O)Nc1cc(NC(=O)c2ccc(N3CCNCC3)cc2)ccc1OCC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.47
ITGA2B P08514 2/20 0.47
ITGA2 P17301 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
NPC1 O15118 4/20 0.44
PTGDR Q13258 1/20 0.43
MAPT P10636 6/20 0.43
KMT2A Q03164 6/20 0.43
MEN1 O00255 5/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 3/20 0.43
HSD17B10 Q99714 3/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477799 0.89 USP28 (0.45) ITGB3ITGA2BITGA2SIRT2SIRT1
Pyridine SCHEMBL8631988 0.87 SIRT2 (0.47) ITGB3ITGA2BITGA2SIRT2SIRT1
SCHEMBL8321319 0.85 ITGB3 (0.51) ITGB3ITGA2BITGA2SIRT2SIRT1
SCHEMBL8318988 0.84 MAPT (0.57) ITGB3ITGA2BITGA2NPC1MAPT
SCHEMBL8320980 0.80 MAPT (0.58) ITGB3ITGA2BITGA2MAPTKMT2A
SCHEMBL8662466 0.78 MAPT (0.61) ITGB3ITGA2BNPC1MAPTKMT2A
Hydrochloric Acid SCHEMBL9409454 0.77 MAPT (0.60) ITGB3ITGA2BITGA2NPC1MAPT
SCHEMBL8661696 0.75 MAPT (0.47) NPC1MAPTKMT2AMEN1SMN1; SMN2
SCHEMBL8322543 0.74 LMNA (0.52) ITGB3ITGA2BNPC1PTGDRMAPT
SCHEMBL8321062 0.73 KIT (0.48) ITGB3ITGA2BITGA2PTGDRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912175-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-09-08 EP disclosed
EP-0922035-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 1999-06-16 EP disclosed
EP-0912175-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1999-05-06 EP disclosed
US-5854245-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-12-29 US disclosed
WO-1998006699-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 1998-02-19 WO disclosed
WO-1998000134-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-01-08 WO disclosed