SCHEMBL8326433

SCHEMBL8326433

N#Cc1ccc(N(Cc2ccc(I)cc2)c2cncnc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.39
POLB P06746 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
AR P10275 1/20 0.34
CYP2A6 P11509 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
STS P08842 1/20 0.33
CTSK P43235 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328066 0.93 CYP19A1 (0.44) CYP19A1POLBCRHBPCRHR2HRH3
SCHEMBL8329428 0.86 MAOA (0.42) CYP19A1POLBCRHBPCRHR2CYP11B1
SCHEMBL8323103 0.86 ESR1 (0.49) CYP19A1CYP11B1CYP11B2
SCHEMBL8325528 0.86 CYP19A1 (0.53) CYP19A1POLBCRHBPCRHR2HRH3
SCHEMBL8324221 0.86 AR (0.45) CYP19A1POLBCRHBPCRHR2AR
SCHEMBL9226442 0.85 CYP11B2 (0.42) CYP19A1POLBCRHBPCRHR2AR
SCHEMBL8324619 0.81 KCNJ1 (0.46) CYP19A1POLBCRHBPCRHR2AR
SCHEMBL8323517 0.81 KCNJ1 (0.46) CYP19A1POLBCRHBPCRHR2AR
SCHEMBL8327043 0.80 CYP19A1 (0.45) CYP19A1STS
SCHEMBL8327702 0.80 CYP19A1 (0.36) CYP19A1POLBHRH3CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed