SCHEMBL8326659

SCHEMBL8326659

COC(=O)C1Cc2c(C)ccc(C)c2N1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
CYP2C19 P33261 1/20 0.45
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
CCKBR P32239 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
PDE5A O76074 4/20 0.36
OPRM1 P35372 1/20 0.35
OGFRL1 Q5TC84 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565447 0.78 KDM4E (0.44) KDM4EHSD17B10ALDH1A1CYP1A2GAA
SCHEMBL6583379 0.74 ALDH1A1 (0.32) KDM4EHSD17B10ALDH1A1CYP1A2CYP2D6
SCHEMBL32677208 0.73 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CYP1A2GAA
SCHEMBL32677091 0.73 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CYP1A2GAA
SCHEMBL32676819 0.73 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CYP1A2GAA
SCHEMBL21739635 0.72 SMYD3 (0.48)
SCHEMBL29015454 0.72 PDE5A (0.38) KDM4EHSD17B10ALDH1A1CYP1A2GAA
SCHEMBL21739383 0.70 KCNH2 (0.33) ALDH1A1TSHRHTT
SCHEMBL8301307 0.69 HSD17B10 (0.39) KDM4EHSD17B10ALDH1A1CYP1A2CYP2D6
SCHEMBL8745451 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866594-A Indole-2-carboxylate derivatives and fungicidal compositions for agricultural or horticultural use containing the derivatives as active component OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1999-02-02 US disclosed
EP-0791582-A1 INDOLE-2-CARBOXYLIC ESTER DERIVATIVES AND AGRICULTURAL AND HORTICULTURAL BACTERIOCIDES CONTAINING THE SAME AS THE ACTIVE INGREDIENT OTSUKA KAGAKU KABUSHIKI KAISHA (JP) 1997-08-27 EP disclosed