SCHEMBL8327210

SCHEMBL8327210

CC(=O)c1ccc(N(Cc2ccc(Br)cc2)c2cncnc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.45
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PYCR1 P32322 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 2/20 0.39
LSS P48449 2/20 0.39
AR P10275 1/20 0.39
GRM5 P41594 1/20 0.38
TSHR P16473 1/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PKM P14618 1/20 0.36
RECQL P46063 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330023 0.79 HTT (0.37) PYCR1KMT2ATSHRHTTSMN1; SMN2
Oxalic Acid SCHEMBL8326149 0.78 AR (0.39) HDAC1HDAC8HDAC6KMT2ALSS
SCHEMBL8325528 0.76 CYP19A1 (0.53) MAOBARTSHRMAOA
SCHEMBL28376324 0.72 ESR1 (0.50) MAOBHDAC1HDAC8HDAC6PYCR1
SCHEMBL10673927 0.70 POLB (0.43) ALDH1A1KDM4EKMT2ALSSGRM5
SCHEMBL17187852 0.69 CES2 (0.62) MAOBMAPTHPGDKMT2ASMN1; SMN2
SCHEMBL20102 0.69 CES2 (0.62) MAOBMAPTHPGDKMT2ASMN1; SMN2
SCHEMBL8327952 0.68 CRHBP (0.47) PYCR1ALDH1A1ARNPSR1
Cyanide SCHEMBL27492933 0.67 RAB9A (0.56) MAOBMAPTHPGDKMT2ASMN1; SMN2
SCHEMBL8328066 0.67 CYP19A1 (0.44) ALDH1A1KDM4EHPGDAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed