Oxalic Acid

Oxalic Acid

SCHEMBL8326149

FC(F)(F)c1ccc(N(Cc2ccc(Br)cc2)c2cncnc2)cc1.O=C(O)C(=O)O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.39
CYP19A1 P11511 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC8 Q9BY41 2/20 0.39
CYP3A4 P08684 1/20 0.36
GCGR P47871 4/20 0.36
GIPR P48546 4/20 0.36
LSS P48449 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
MTOR P42345 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HIF1A Q16665 1/20 0.34
EPAS1 Q99814 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327210 0.78 MAOB (0.45) ARHDAC1HDAC6HDAC8LSS
SCHEMBL8329070 0.77 MMP1 (0.45) ARCYP19A1
SCHEMBL8330023 0.73 HTT (0.37) CYP19A1CYP3A4MEN1KMT2A
SCHEMBL6718505 0.72 MEN1 (0.43) HDAC1HDAC6HDAC8LSSMTOR
SCHEMBL8325528 0.72 CYP19A1 (0.53) ARCYP19A1
SCHEMBL4590779 0.69 GBA1 (0.44) ARHDAC1HDAC6HDAC8MTOR
SCHEMBL28376324 0.69 ESR1 (0.50) CYP19A1HDAC1HDAC6HDAC8
SCHEMBL10673927 0.67 POLB (0.43) CYP19A1CYP3A4LSSMEN1KMT2A
SCHEMBL6171116 0.66 CYP3A4 (0.46) HDAC1HDAC6HDAC8CYP3A4KMT2A
SCHEMBL8327952 0.65 CRHBP (0.47) ARCYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed