SCHEMBL8327952

SCHEMBL8327952

O=[N+]([O-])c1ccc(CN(c2ccc([N+](=O)[O-])cc2)c2cncnc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
AR P10275 10/20 0.45
POLB P06746 1/20 0.45
CYP19A1 P11511 2/20 0.45
PYCR1 P32322 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326188 0.93 CYP19A1 (0.55) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8323939 0.93 AR (0.49) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8327171 0.93 CRHBP (0.42) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8327623 0.93 ALDH1A1 (0.50) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8329070 0.90 MMP1 (0.45) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8323517 0.90 KCNJ1 (0.46) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL8324619 0.90 KCNJ1 (0.46) CRHBPCRHR2ARPOLBCYP19A1
SCHEMBL5843018 0.78 CRHBP (0.64) CRHBPCRHR2ARALDH1A1CYP1A2
SCHEMBL8327373 0.77 ALDH1A1 (0.61) CRHBPCRHR2POLBCYP19A1ALDH1A1
SCHEMBL8327951 0.73 SLC29A1 (0.41) POLBALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed